Keywords imatinib mesylate;enaminone;aminopyrimidine;coupling reaction;Heteroarylamine;aryl halid;copper catalysis;hydrazine hydrate reduction;total synthesis;

• 甲磺酸伊马替尼;烯胺酮;嘧啶胺;偶联反应;芳香杂环胺;芳基卤化物;铜催化;水合肼还原;全合成;